SCH-202,596
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| Clinical data | |
|---|---|
| ATC code | none |
| Identifiers | |
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| CAS Number | 196615-89-1 |
| PubChem (CID) | 11758032 |
| IUPHAR/BPS | 6128 |
| Chemical and physical data | |
| Formula | C25H22Cl2O12 |
| Molar mass | 585.340 g/mol |
| 3D model (Jmol) | Interactive image |
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SCH-202,596 is a natural product which is a metabolite derived from an Aspergillus fungus. It acts as a selective non-peptide antagonist for the receptor GAL-1, which is usually activated by the neuropeptide galanin. SCH-202,596 is used for scientific research into this still little characterised receptor subtype.[1][2]
References
- ↑ Min C, et al. A New Fungal Metabolite, Sch 202596, with Inhibitory Activity in the Galanin Receptor GALR1 Assay. Tetrahedron Letters 1997; 38(35):6111–6114. doi:10.1016/S0040-4039(97)01385-3
- ↑ Katoh T, et al. Synthetic studies on Sch 202596, an antagonist of the galanin receptor subtype GalR1: an efficient synthesis of (±)-geodin, the spirocoumaranone part of Sch 202596. Tetrahedron 2002; 58(7):1289–1299.
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